FIELD: medicine; pharmaceutics.
SUBSTANCE: invention relates to a compound of formula III or a pharmaceutically acceptable salt thereof, where each R1, R2 is independently selected from the group consisting of hydrogen and C1-6 alkyl; m = 1, 2, 3 or 4.
EFFECT: compound of formula III is a neurokinin-1 receptor antagonist, can be used to treat diseases associated with the neurokinin-1 receptor, for example for treating vomiting, nausea, depression or anxiety in a patient, and also allows to avoid haemolytic effects of drugs and reduce side effects of drug administration.
4 cl, 1 dwg, 8 tbl, 18 ex
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