CONJUGATES AND SMALL MOLECULES, INTERACTING WITH CD16a RECEPTOR Russian patent published in 2014 - IPC C07D281/16 C07D495/14 C07K14/555 C12P21/08 A61K31/554 A61K31/5517 A61K38/02 A61P35/00 A61P37/00 

Abstract RU 2519546 C1

FIELD: chemistry.

SUBSTANCE: compounds can be applied for treatment of oncologic and autoimmune diseases. Invention also characterises method of obtaining conjugates, pharmaceutical composition and medication, which contains modified proteins. In general formulae 1 or 2 , R1 is selected from the group representing (CH3)2N-,

R2 is selected from the group representing where R3 as terminal substituent represents -NH2, or and R4 represents H or C1-C3alkyl.

EFFECT: novel compounds possess affinity for CD16a receptor.

18 cl, 20 dwg, 3 tbl, 19 ex

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RU 2 519 546 C1

Authors

Demin Aleksandr Viktorovich

Tkachenko Sergej Evgen'Evich

Dates

2014-06-10Published

2013-01-16Filed