FIELD: chemistry.
SUBSTANCE: invention relates to 2-{4-amino-2-[(3-chloro-4-methoxy-5-methylpyridin-2-yl)methyl]-2,7-dihydro-6-thia-1,2,3,5-tetraazabenzo[cd]azulen-8-yl}-N-methylacetamide and its salts, such as hydrobromide, hydrochloride, methane sulfonate, ethane-1,2-disulfonate. The invention also relates to a medication and a pharmaceutical composition based on the said compound and its salts for inhibition of ATP-ase activity of HSP90.
EFFECT: novel compound and its salts, which can be applied in medicine for cancer treatment, are obtained.
23 cl, 10 ex
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Authors
Dates
2014-06-27—Published
2010-02-24—Filed