FIELD: medicine, pharmaceutics.
SUBSTANCE: invention refers to a diagnostic and therapeutic agent which is a bombesin analogue peptide antagonist conjugate having the general formula (I), [A-(B)n]x-C, wherein A represents a metal chelator containing at least one radionuclide metal, B represents a spacer bound to N terminal C, or a covalent bond, and C represents a bombasin analogue peptide antagonist, wherein additionally x represents an integer 1 to 3, and n represents an integer 1 to 6.
EFFECT: preparing the therapeutic agent representing the bombesin analogue peptide antagonist conjugate.
17 cl, 12 dwg, 1 tbl, 13 ex
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