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(19)

RU

(11)

2 821 944

(13)

C2

(51)

IPC

C07K7/06(2006-01-01)

A61K103/00(2006-01-01)

A61K103/30(2006-01-01)

A61K51/08(2006-01-01)

A61P35/00(2006-01-01)

C07B59/00(2006-01-01)

(21) (22)

Application

2019119378, 2013-09-25

(24)

Start date

2013-09-25

(22)

Actual filing date

2013-09-25

(45)

Published

2024-06-28

(72)

Inventor

Maina-Nock, TheodosiaNock, Berthold, ArturDe Jong Hendriks, Marion

(73)

Holder

Advanced Accelerator Applications Usa, Inc.

GRPR ANTAGONISTS FOR DETECTING, DIAGNOSING AND TREATING GRPR-POSITIVE ONCOLOGICAL DISEASE Russian patent published in 2024 - IPC C07K7/06 A61K103/00 A61K103/30 A61K51/08 A61P35/00 C07B59/00 

Abstract RU 2821944 C2

FIELD: medicine.

SUBSTANCE: present invention relates to the field of diagnosing and treating oncological diseases, specifically to a compound having a structure

,

here M is 177Lu or 68Ga. Invention also relates to a medicinal agent and a therapeutic composition based on said compound.

EFFECT: invention provides high degree of capture and retention of diagnostic and therapeutic radioactive label selectively with respect to both primary and metastatic GRPR+ oncological disease.

6 cl, 8 dwg, 1 ex

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RU 2 821 944 C2

Authors

Maina-Nock, Theodosia

Nock, Berthold, Artur

De Jong Hendriks, Marion

Dates

2024-06-28—Published

2013-09-25—Filed

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