CYCLIC OCTAPEPTIDE, RADIOPHARMACEUTICAL AGENT BASED THEREON AND METHOD OF USING RADIOPHARMACEUTICAL AGENT TO PRODUCE MEDICINAL (PHARMACEUTICAL) AGENTS FOR TREATING NEOPLASMS EXPRESSING SOMATOSTATIN RECEPTORS Russian patent published in 2014 - IPC C07K7/06 C07K14/655 A61K38/08 A61K38/31 A61K51/08 

Abstract RU 2528414 C1

FIELD: chemistry.

SUBSTANCE: radiopharmaceutical agent of formula (Ia) or (Ib) , is a cyclic octapeptide complex which contains a chelating group with radionuclides 111In, 90Y, 177Lu. The radiopharmaceutical agent can be used to produce medicinal agents for radionuclide therapy of neoplasms which express somatostatin receptors. X is a chelating agent.

EFFECT: improved properties.

2 cl, 1 dwg, 2 tbl, 6 ex

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RU 2 528 414 C1

Authors

Nazarenko Anna Borisovna

Voloznev Lev Vasil'Evich

Grinin Maksim Gennad'Evich

Dates

2014-09-20Published

2013-01-25Filed