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2 534 525

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IPC

C07D339/04(2006-01-01)

A61K31/385(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2013143268/04, 2013-09-24

(24)

Start date

2013-09-24

(22)

Actual filing date

2013-09-24

(45)

Published

2014-11-27

(72)

Inventor

Fedorov Sergej NikolaevichKuz'Mich Aleksandra SergeevnaPolonik Sergej GeorgievichDyshlovoj Sergej Anatol'EvichShubina Larisa KimovnaRakitin Oleg AlekseevichOgurtsov Vladimir Anatol'Evich

(73)

Holder

Federal'Noe Gosudarstvennoe Bjudzhetnoe Uchrezhdenie Nauki Tikhookeanskij Institut Bioorganicheskoj Khimii Im. G.B. Eljakova Dal'Nevostochnogo Otdelenija Rossijskoj Akademii Nauk Dvo Ran)

GLYCOSIDE DERIVATIVES OF 1,2-DITHIOL-3-THIONE OR 1,2-DITHIOL-3-ONE AND PHARMACEUTICAL PRODUCTS BASED ON THEM Russian patent published in 2014 - IPC C07D339/04 A61K31/385 A61P35/00

Abstract RU 2534525 C9

FIELD: biotechnology.

SUBSTANCE: invention relates to glycosidic derivatives of 1,2-dithiole-3-thione or 1,2-dithiol-3-one of formula 1 , where R₁=S or O; R₂ is a residue of per-O-acetyl D-glucose, per-O-acetyl D-galactose, per-O-acetyl D-mannose, per-O-acetyl D-xylose, per-O-acetyl L-arabinose, per-O-acetyl-D-maltose or D-glucose, which can be used against cancerous diseases.

EFFECT: new bioactive compounds with cancerous preventive action and pharmaceutical products based on them are proposed, which display the cancerous preventive effect in non-cytotoxic concentrations.

2 cl, 4 ex, 5 tbl

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RU 2 534 525 C9

Authors

Fedorov Sergej Nikolaevich

Kuz'Mich Aleksandra Sergeevna

Polonik Sergej Georgievich

Dyshlovoj Sergej Anatol'Evich

Shubina Larisa Kimovna

Rakitin Oleg Alekseevich

Ogurtsov Vladimir Anatol'Evich

Dates

2014-11-27—Published

2013-09-24—Filed