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2 547 835

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IPC

C07D401/04(2006-01-01)

C07D491/06(2006-01-01)

C07D471/04(2006-01-01)

C07D487/04(2006-01-01)

A61K31/4985(2006-01-01)

A61K31/53(2006-01-01)

A61P31/00(2006-01-01)

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Application

2014108753/04, 2014-03-06

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Start date

2014-03-06

(22)

Actual filing date

2014-03-06

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Published

2015-04-10

(72)

Inventor

Chupakhin Oleg NikolaevichCharushin Valerij NikolaevichKotovskaja Svetlana KonstantinovnaRusinov Vladimir LeonidovichUlomskij Evgenij NartsissovichBykov Vladimir NikolaevichStepanov Aleksandr ValentinovichChepur Sergej ViktorovichLebedeva Irina KirillovnaTsikarishvili Georgij VarlamovichKurpjakova Anna Fedorovna

(73)

Holder

Federal'Noe Gosudarstvennoe Bjudzhetnoe Uchrezhdenie Nauki Institut Organicheskogo Sinteza Im. I.Ja. Postovskogo Ural'Skogo Otdelenija Rossijskoj Akademii Nauk

AZOLOAZINE SALTS OF FLUOROQUINOLONES, POSSESSING ANTIBACTERIAL AND ANTIVIRAL ACTION Russian patent published in 2015 - IPC C07D401/04 C07D491/06 C07D471/04 C07D487/04 A61K31/4985 A61K31/53 A61P31/00

Abstract RU 2547835 C1

FIELD: chemistry.

SUBSTANCE: invention relates to azoloazine salts of compounds of a fluoroquinolone line of formulae 4a-c , 5a-c , 7a-b and 8a-b , possessing antibacterial and antiviral properties. The claimed compounds can be applied for the creation of a medication for the emergency prevention and treatment of infections, caused by pathogens of both the bacterial and viral origin, including especially dangerous ones. In general formulae 4 and 5 R=CH₃, R₁=C₂H₅; R=H, R₁=C₂H₅; R=C₂H₅, R₁=cyclo-C₃H_7,in formulae 7 and 8 R=H (7a, 8a); R=CH₃ (7b, 8b).

EFFECT: increased efficiency of the compound application.

8 tbl, 2 ex

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RU 2 547 835 C1

Authors

Chupakhin Oleg Nikolaevich

Charushin Valerij Nikolaevich

Kotovskaja Svetlana Konstantinovna

Rusinov Vladimir Leonidovich

Ulomskij Evgenij Nartsissovich

Bykov Vladimir Nikolaevich

Stepanov Aleksandr Valentinovich

Chepur Sergej Viktorovich

Lebedeva Irina Kirillovna

Tsikarishvili Georgij Varlamovich

Kurpjakova Anna Fedorovna

Dates

2015-04-10—Published

2014-03-06—Filed