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RU

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2 839 407

(13)

C1

(51)

IPC

C07D487/04(2006-01-01)

A61K31/519(2006-01-01)

A61P31/12(2006-01-01)

A61P31/14(2006-01-01)

(21) (22)

Application

2024121106, 2024-07-23

(24)

Start date

2024-07-23

(22)

Actual filing date

2024-07-23

(45)

Published

2025-04-30

(72)

Inventor

Mukhin Evgenij MikhajlovichSavateev Konstantin ValerevichKotovskaya Svetlana KonstantinovnaRusinov Vladimir LeonidovichVaraksin Mikhail ViktorovichPyankov Oleg ViktorovichShipovalov Andrej VladimirovichKudrov Gleb AleksandrovichZajkovskaya Anna VladimirovnaSkarnovich Maksim Olegovich

(73)

Holder

Federalnoe Gosudarstvennoe Avtonomnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniya Federalnyj Universitet Imeni Pervogo Prezidenta Rossii B.N. Eltsina"Federalnoe Byudzhetnoe Uchrezhdenie Nauki Nauchnyj Tsentr Virusologii I Biotekhnologii Federalnoj Sluzhby Po Nadzoru V Sfere Zashchity Prav Potrebitelej I Blagopoluchiya Cheloveka

ETHYL ESTER OF 2-(ADAMANTAN-1-yl)-3-BROMO-7-OXO-4,7-DIHYDROPYRAZOLO[1,5-a]PYRIMIDINE-6-CARBOXYLIC ACID, HAVING ANTIVIRAL ACTION ON SARS-CoV-2 CORONAVIRUS Russian patent published in 2025 - IPC C07D487/04 A61K31/519 A61P31/12 A61P31/14 

Abstract RU 2839407 C1

FIELD: chemistry.

SUBSTANCE: invention relates to ethyl ester of 2-(adamantan-1-yl)-3-bromo-7-oxo-4,7-dihydropyrazolo[1,5-a]pyrimidine-6-carboxylic acid 3,

having a pronounced inhibitory effect action on coronavirus SARS-CoV-2, strain hCoV-19/Russia/Vologda-171613-1208/2020.

EFFECT: obtaining a novel compound which can be used against coronavirus SARS-CoV-2, strain hCoV-19/Russia/Vologda-171613-1208/2020.

1 cl, 1 dwg, 1 tbl

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RU 2 839 407 C1

Authors

Mukhin Evgenij Mikhajlovich

Savateev Konstantin Valerevich

Kotovskaya Svetlana Konstantinovna

Rusinov Vladimir Leonidovich

Varaksin Mikhail Viktorovich

Pyankov Oleg Viktorovich

Shipovalov Andrej Vladimirovich

Kudrov Gleb Aleksandrovich

Zajkovskaya Anna Vladimirovna

Skarnovich Maksim Olegovich

Dates

2025-04-30—Published

2024-07-23—Filed

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