PHARMACEUTICAL COMPOSITION CONTAINING QUINOLINE DERIVATIVE Russian patent published in 2015 - IPC A61K31/47 A61K47/32 A61K47/36 A61K47/38 A61P35/00 

Abstract RU 2548673 C2

FIELD: medicine.

SUBSTANCE: invention refers to a pharmaceutical composition containing a compound presented by formula (I) , wherein R1 represents a hydrogen atom, C1-6 alkyl group or C3-8 cycloalkyl group; while R2 represents a hydrogen atom or a methoxyl group, or its pharmaceutically acceptable salt, or solvate; and alkaline earth carbonate, wherein the content of the compound presented by formula (I), or its salt or solvate makes 0.25 to 50 wt %, and the content of alkaline earth carbonate makes 1 to 60 wt % in relation to total weight of the composition, respectively.

EFFECT: composition exhibits excellent solubility; it is storage-stable or even long-term storage-stable, and applicable as a preventive or therapeutic agent for treating a tumour.

10 cl, 7 dwg, 10 tbl, 19 ex

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RU 2 548 673 C2

Authors

Bando Masasi

Dates

2015-04-20Published

2010-08-16Filed