FIELD: chemistry.
SUBSTANCE: invention relates to synthetic biologically active heterocyclic substances having antagonist activity on purinoreceptors and which are products of modifying pyridoxin, particularly n-(1,5-dihydro-3-R-8-methyl-9-hydroxy-[1,3]dioxepino[5,6-c]pyridinyl-6-azo)phenyl sulphonic acid and salt forms thereof of general formula I 
, where is selected from: a hydrogen atom, ethyl, heptyl or octyl.
EFFECT: compounds of the given formula have high antagonist activity on purinoreceptors and can be used in medicine and veterinary.
2 tbl, 5 ex
| Title | Year | Author | Number |
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