FIELD: chemistry.
SUBSTANCE: invention relates to synthetic biologically active substances of the heterocyclic series, having anticholinesterase activity, and is a product of modification of pyrodoxine acetals, specifically 1,5-dihydro-3-R1-3-R2-7,8-dimethyl-9-dimethylcarbamoyloxy-[1,3]dioxepino[5,6-c]pyridinium bromide of general formula I, where R1 is a hydrogen atom or a methyl, R2 is selected from: methyl, ethyl, propyl, iso-propyl, tert-butyl, heptyl, octyl or (1-methyldecyl). The compounds of formula (I) 
have high anticholinesterase activity and can be used in medicine and veterinary.
EFFECT: high activity of the compounds.
2 tbl, 11 ex
| Title | Year | Author | Number |
|---|---|---|---|
| ANTIBACTERIAL COMPOUNDS BASED ON SULPHANILIC ACID AND PYRIDOXINE | 2012 |
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| PHOSPHONIUM SALTS ON BASIS OF PYRIDOXINE DERIVATIVES | 2011 |
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|
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| INHIBITORS OF FORMATION OF GLYCATION END PRODUCTS BASED ON AZO-DERIVATIVE PHENYLSULPHONIC ACIDS | 2016 |
|
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| QUATERNARY AMMONIUM SALTS BASED ON DERIVATIVES OF VITAMIN B6 | 2015 |
|
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| ANTIBACTERIAL AGENTS BASED ON QUATERNARY AMMONIUM SALTS | 2014 |
|
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| PYRIDOXINE DERIVATIVE-BASED BETA-ADRENERGIC BLOCKING AGENTS | 2014 |
|
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| AZO DERIVATIVES OF 5-AMINOSALICYLIC ACID, CAPABLE OF INHIBITING FORMATION OF END PRODUCTS OF GLYCATION | 2024 |
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RU2837878C1 |
