N-SULPHATED OLIGOSACCHARIDES ACTIVATING FGF RECEPTORS, PRODUCING AND USING THEM IN THERAPY Russian patent published in 2015 - IPC A61K31/737 C07H13/04 C07H13/12 C07H15/203 C08B37/00 

Abstract RU 2559629 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: present invention refers to oligosaccharides activating FGF receptors, and applying them in medicine of formula (I):

, wherein R2 represents -O-alkyl or monosaccharide of formula , R represents alkyl, R3 is disaccharide of formula , R5 is disaccharide of formula , R7 represents OH or disaccharide of formula , R1, R4, R6 and R8 represents -OSO3- or OH, but other than OH-groups simultaneously, R9 represents OH, -O-alkyl or disaccharide of formula , R10 represents -O-alkyl provided R9 represents OH or -O-alkyl if R2 is monosaccharide of formula (II), R7 represents disaccharide of formula (VI) if R2 represents -O-alkyl.

EFFECT: there are presented new substances stimulating angiogenesis.

24 cl, 9 ex

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Authors

Djushossua Filipp

Fon P'Er

Fruadbiz Aleksandr

Dates

2015-08-10Published

2010-08-12Filed