CRYSTALLINE β-MODIFICATION OF 2,3-BIS-(HYDROXYMETHYL)QUINOXALINE-N,N'-DIOXIDE, METHOD OF THEREOF OBTAINING AND THEREOF-BASED PHARMACEUTICAL COMPOSITION Russian patent published in 2015 - IPC C07D241/52 A61K31/4985 A61P31/04 

Abstract RU 2563256 C1

FIELD: chemistry.

SUBSTANCE: invention relates to crystalline β-modification of 2,3-bis-(hydroxymethyl)quinoxaline-N,N'-dioxide (dioxidine), method of its obtaining and its application for preparation of pharmaceutical composition, possessing antimicrobial, antibacterial and bactericidal activity.

EFFECT: crystalline dioxidine β-modification possesses increased antimicrobial, antibacterial and bactericidal activity in comparison with activity of initial dioxidine substance.

3 cl, 8 dwg, 4 tbl, 4 ex

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RU 2 563 256 C1

Authors

Shabatin Vladimir Petrovich

Vernaja Ol'Ga Ivanovna

Semenov Aleksandr Mikhajlovich

Shabatina Tat'Jana Igorevna

Dates

2015-09-20Published

2014-04-11Filed