FIELD: medicine, pharmaceutics.
SUBSTANCE: claimed invention relates to novel cyclopentyl- and cycloheptylpyrazole derivatives of formula I, where A and R1-R4 are determined in formula of invention, or their pharmaceutically acceptable salts. Invention also relates to pharmaceutical composition containing them and application of claimed compounds.
EFFECT: compounds of formula are modulators of FXR activity.
14 cl, 20 ex
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Authors
Dates
2015-11-10—Published
2011-03-21—Filed