NOVEL CONSTRUCTIONS OF TRANSPORTERS AND CONJUGATE MOLUCELES WHICH ARE TRASPORTERS OF CARGO-MOLECULES Russian patent published in 2015 - IPC C07K14/16 A61K39/00 

Abstract RU 2570632 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: invention relates to field of biotechnology. Also disclosed conjugate molecules, which are transporters of cargo-molecules, in particular, conjugates of novel constructions of transporters with cargo-fragment, for example, with proteins or peptides, nucleic acids, cytotoxic agents, organic molecules, etc. Also described pharmaceutical compositions, which contain said conjugates and methods of treatment and application with application of said constructions of transporters. Claimed group of inventions can be applied in medicine.

EFFECT: novel constructions of transporters of general formula (I) D1LLLxDm(LLLyDn)a and their versions are described.

18 cl, 22 dwg, 6 tbl, 29 ex

Similar patents RU2570632C2

Title Year Author Number
EFFECTIVE TRANSPORT INTO LEUKOCYTES 2009
  • Kristof Bonni
RU2558240C2
NOVEL MOLECULE INHIBITORS OF JNK 2011
  • Bonni Kristof
RU2570417C2
COMPOSITIONS AND METHODS FOR DIAGNOSTICS AND TREATMENT OF TUMOUR 2010
  • Dehnnis Mark
  • Polakis Pol
  • Rubinfeld Bonni
RU2563359C2
METHODS AND COMPOSITION FOR INHIBITION OF HIV-1 MULTIPLICATION 2001
  • Gol'Dshtejn Gideon
RU2275379C2
FUSION CONSTRUCTION CONTAINING CELL PENETRATING PEPTIDE, POLYEPITOPE AND TLR PEPTIDE AGONIST, INTENDED FOR TREATMENT OF CANCER 2017
  • Derouazi Madiha
  • Belnoue Elodie
RU2807135C2
COMBINATION OF AN IMMUNE CHECKPOINT MODULATOR AND A COMPLEX CONTAINING A CELL-PENETRATING PEPTIDE, A CARGO MOLECULE, AND A TLR PEPTIDE AGONIST, FOR APPLICATION IN MEDICINE 2017
  • Derouazi Madiha
  • Belnoue Elodie
RU2769314C1
COMBINATION OF IMMUNE CHECKPOINT MODULATOR AND COMPLEX CONTAINING CELL-PENETRATING PEPTIDE, CARGO MOLECULE, AND TLR PEPTIDE AGONIST FOR MEDICAL USE 2017
  • Deruazi Madikha
  • Belnu Elodi
RU2748378C2
PEPTIDE VECTORS 2004
  • Dong Chzhen Ksin
  • Shen Jilana
  • Komstok Dzhinn Mehri
  • Kim San Kh.
RU2361876C2
GLYCATED PEPTIDE GLP-1 2009
  • Kadzikhara, Jasukhiro
  • Tsjudzi, Takasi
  • Sakamoto, Izumi
  • Nambu, Juri
  • Khajasi, Naokhiro
  • Isii, Kazujuki
  • Fukae, Kazukhiro
  • Tezuka, Katsunari
  • Asai, Khiroaki
RU2543157C2
OBTAINING OF COMPLEXES OF NUCLEIC ACIDS AND CATIONIC COMPONENTS CROSS SEWED BY DISULFIDE BONDS INTENDED FOR TRANSFECTION AND IMMUNOSTIMULATION 2011
  • Baumkhof Patrik
  • Foss Zenke
  • Kramps Tomas
  • Kallen Karl-Jozef
RU2575603C2

RU 2 570 632 C2

Authors

Kristof Bonni

Dates

2015-12-10Published

2009-12-22Filed