NEUROPROTECTIVE AGENT BASED ON BIS{2-[(2E)-4-HYDROXY-4-OXOBUT-2-ENOYLOXY]-N,N-DIETHYLETHANAMINE}BUTANDIOATE Russian patent published in 2016 - IPC A61K31/221 A61K31/194 A61P25/00 

Abstract RU 2588365 C1

FIELD: medicine; pharmaceuticals.

SUBSTANCE: invention relates to a novel neuroprotective agent based on bis{2-[(2E)-4-hydroxy-4-oxobut-2-enoyloxy]-N,N-diethylethanamine}butandioate (I). Shows neuroprotective action of compound as active substance included in drug on hypoxia model, it has antiasthenic, nootropic and actoprotective action. Compound is low toxic, by efficiency is comparable with used in practice taken separately nootropic, actoprotective, antihypoxic preparations.

EFFECT: said properties enable to assume that bis{2-[(2E)-4-hydroxy-4-oxobut-2-enoyloxy]-N,N-diethylethanamine}butandioate can be used in medicine.

1 cl, 1 dwg, 6 tbl, 5 ex

I

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RU 2 588 365 C1

Authors

Okovityj Sergej Vladimirovich

Shustov Evgenij Borisovich

Bolotova Vera Tsezarevna

Titovich Irina Aleksandrovna

Dates

2016-06-27Published

2015-05-19Filed