METHOD OF PRODUCING CYCLOPROPANE DERIVATIVES Russian patent published in 2016 - IPC C07D321/10 

Abstract RU 2593202 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a compound of formula (5): wherein n represents 0, and R11 is hydroxyl, or its tautomer, racemate or stereoisomer thereof, which is intermediate compound for producing cyclopropane particularly 2-amino-9-[[1S,2R)-1,2-bis (hydroxymethyl)cyclopropyl]methyl]-1,9-purine-6-one, which has antiviral activity, as well as method for preparing them.

EFFECT: obtaining cyclopropane derivatives.

11 cl

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RU 2 593 202 C2

Authors

Kiss Eleonora

Blomsma Ervin

De Brejn Serzh

Litens E.J.N. Remi

Dates

2016-08-10Published

2011-11-10Filed