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(19)

(11)

2 401 833

(13)

(51)

IPC

C07D253/75(2006-01-01)

A61K31/53(2006-01-01)

A61P31/18(2006-01-01)

(21) (22)

Application

2007108539/04, 2005-08-10

(24)

Start date

2005-08-10

(22)

Actual filing date

2005-08-10

(45)

Published

2010-10-20

(72)

Inventor

Zhanssen Pol' Adrian JanKhornart Dzhorzh Zhozef KorneliusKilonda AmuriKheres JanLevi Paulus JoannesDe Zhonzh Mark ReneDajer Frederik Frans DezireVinkers Khendrik MartenKojmans Ljus'En Marija Khenrikus

(73)

Holder

Janssen Farmatsevtika N.V.

1,2,4-TRIAZINE-6-ONE DERIVATIVES, INHIBITING HIV Russian patent published in 2010 - IPC C07D253/75 A61K31/53 A61P31/18

Abstract RU 2401833 C2

FIELD: medicine, pharmaceutics.

SUBSTANCE: described are novel derivatives of 1,2,4-triazine-6-one of general formula (I) or their pharmaceutically acceptable acid-additive salts, or stereochemically isomeric forms, where rings A and B represent phenyl; values of other radicals are given in formula of invention.

EFFECT: development of efficient method of obtaining composition and application of novel compounds for treatment or prevention of HIV-infection.

22 cl, 2 tbl, 6 ex

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RU 2 401 833 C2

Authors

Zhanssen Pol' Adrian Jan

Khornart Dzhorzh Zhozef Kornelius

Kilonda Amuri

Kheres Jan

Levi Paulus Joannes

De Zhonzh Mark Rene

Dajer Frederik Frans Dezire

Vinkers Khendrik Marten

Kojmans Ljus'En Marija Khenrikus

Dates

2010-10-20—Published

2005-08-10—Filed