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2 593 998

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IPC

C07D307/78(2006-01-01)

A61K31/343(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2015124722/04, 2015-06-23

(24)

Start date

2015-06-23

(22)

Actual filing date

2015-06-23

(45)

Published

2016-08-10

(72)

Inventor

Fedorov Aleksej YurevichGracheva Yuliya AleksandrovnaVojtovich Yuliya ValerevnaSvirshshevskaya Elena ViktorovnaKuznetsov Andrej Grigorevich

(73)

Holder

Federalnoe Gosudarstvennoe Avtonomnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniya Gosudarstvennyj Universitet Im. N.I. Lobachevskogo"

1',2',3'-TRIMETOXIBENZO[5',6:5,4]-1H-6,7-DIHYDROCYCLOGEPTA[3,2-f]BENZOFURAN DERIVATIVE AND ITS APPLICATION Russian patent published in 2016 - IPC C07D307/78 A61K31/343 A61P35/00

Abstract RU 2593998 C1

FIELD: chemistry.

SUBSTANCE: invention relates to novel derivatives of 1′,2′,3′-trimetoxibenzo[5′,6′:5,4]-1H-6,7-dihydrocyclogepta[3,2-f]benzofuran represented by the general formula, where R is the substitute, R=CH₂OH, CH(CH₃)OH, CH₂CH₂OH, CH₂OAc; X is the functional group, X=O, OH, as well as to the use of these compounds as an active component of anti-tumour medicine for treating oncological diseases.

EFFECT: technical result is the increase of activity at inhibition of tumour cells proliferation.

9 cl, 2 dwg

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RU 2 593 998 C1

Authors

Fedorov Aleksej Yurevich

Gracheva Yuliya Aleksandrovna

Vojtovich Yuliya Valerevna

Svirshshevskaya Elena Viktorovna

Kuznetsov Andrej Grigorevich

Dates

2016-08-10—Published

2015-06-23—Filed