AZAINDAZOLE OR DIAZAINDAZOLE DERIVATIVES AS MEDICINE Russian patent published in 2016 - IPC C07D471/04 C07D487/04 A61K31/437 A61K31/4985 A61P35/00 A61P25/28 

Abstract RU 2600976 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a compound of general formula (I) or a pharmaceutically acceptable salt thereof, in which radicals and symbols assume values given in patent claim. Compound of formula (I) is a kinase inhibitor, such as ALK Abl and/or c-Src.

EFFECT: invention also relates to its use as a drug for treating cancer, inflammation and neurodegenerative diseases, such as Alzheimer's disease, to its use as an inhibitor of said kinases, to a pharmaceutical composition containing said compound, and to methods of its production.

16 cl, 20 tbl, 35 ex

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RU 2 600 976 C2

Authors

Kalun El Bakhir

Bedzhegelal Karim

Rabo Remi

Kryuzinski Anna

Shmitt Filipp

Peres Mishel

Raje Nikolya

Dates

2016-10-27Published

2012-01-27Filed