CRYSTAL HAVING CRYSTAL HABIT, AND PHARMACEUTICAL COMPOSITION PREPARED BY TREATMENT OF SAID CRYSTAL Russian patent published in 2016 - IPC C07D409/06 A61K31/4178 A61P31/10 

Abstract RU 2603963 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a luliconazole crystal presented by formula, wherein crystal has such a crystal habit, that (021) plane is its characteristic plane of crystal growth, in which I(021) in relation to total I(001), I(100), I(10-1), I(011), I(110), I(11-1), I(10-2), I(11-2), I(020), I(021), I(20-2), I(121), I(013), I(11-3) and I(221) is not less than 1/3, provided that relative to diffraction peaks, detected in range of 2θ=5-35° in x-ray powder diffraction using CuKα radiation, integral intensities of diffraction peaks, which correspond to (001), (100), (10-1), (011), (110), (11-1), (10-2), (11 -2), (020), (021), (20-2), (121), (013), (11-3) and (221) planes are designated as I(001), I(100), I(10-1), I(011), I(110), I(11-1), I(10-2), I(11-2), I(020), I(021), I(20-2), I(121), I(013), I(11-3) and I(221) respectively .

EFFECT: invention aims at providing means to improve solubility of luliconazole.

8 cl, 6 dwg, 4 tbl, 4 ex

Similar patents RU2603963C2

Title Year Author Number
NEW CRYSTALS OF URACIL COMPOUND 2016
  • Fukuoka, Masayoshi
RU2686722C1
CRYSTALS 2010
  • Itou Khidejuki
  • Nakamiti Kodzi
  • Tosaka Takasi
RU2556206C2
STABLE CRYSTALLINE FORM OF TYPIRACYL HYDROCHLORIDE AND METHOD FOR ITS CRYSTALLIZATION 2014
  • Kadzuno Khideki
  • Mutsumi Tomonobu
RU2640417C2
AZABICYCLIC COMPOUND CRYSTALS 2016
  • Uno, Takao
RU2697521C2
CRYSTALLINE POLYMORPHYL OF 4-[5-(PYRIDINE-4-YL)-1H-1,2,4-TRIAZOL-3-YL]-PYRIDINE-2-CARBONITRILE AND METHOD OF ITS OBTAINING 2013
  • Ivabuti Josiyuki
  • Miyata Satikho
  • Sato Takakhiro
  • Uda Dzunitiro
  • Kandou Takamitsu
  • Inoue Tadasi
  • Nakano Khiroyuki
RU2639149C2
CRYSTALLINE FORMS OF TIGECYCLINE AND METHOD FOR PREPARING THEM 2006
  • Krishnan Lalita
  • Deshmukh Sabodkh S.
  • Khadfild Ehntoni
  • Khuang Dzhejms V.
  • Ku Manching Sherri
RU2478612C2
STABLE CRYSTALLINE FORM OF TIPIRACIL HYDROCHLORIDE AND METHOD FOR ITS CRYSTALLIZATION 2014
  • Kadzuno Khideki
  • Mutsumi Tomonobu
RU2674441C1
SALT OF MU-OPIOID RECEPTOR (MOR) AGONIST, CRYSTAL FORM I OF ITS FUMARATE SALT, AND THEIR PRODUCTION METHOD 2018
  • Wang, Lin
  • Wang, Likun
RU2779119C2
SALT OF PYRAZOLOQUINOLINE DERIVATIVE AND CRYSTAL THEREOF 2014
  • Odzaki Sunsuke
RU2655171C2
DIMETHYLAMINOCHELIOLIDE FUMARATE HYDRATE AND METHOD FOR PREPARATION THEREOF, AND USE THEREOF 2020
  • Li, Chzhunkhua
  • Gun, Tszyunbo
  • Khou, Baokhun
  • Vu, Sungu
  • Chen, Yue
  • Tsyu, Chuantszyan
  • Chzhu, Sinkhua
  • Tsi, Tsze
  • Van, Gujyan
RU2824144C1

RU 2 603 963 C2

Authors

Masuda Takaaki

Dates

2016-12-10Published

2012-11-02Filed