AGENT FOR REDUCTION OF GLUTAMATE-INDUCED APOPTOSIS AND INHIBITION OF NMDA-RECEPTOR, POSSESSING IMMUNOMODULATORY ACTION, FOR TREATING NERVOUS SYSTEM DISORDERS, EFFECTS OF CRANIOCEREBERAL INJURY AND ISCHEMIC AND HEMORRHAGIC STROKE Russian patent published in 2016 - IPC A61K31/7068 A61K31/13 A61K47/48 A61P9/10 A61P25/00 

Abstract RU 2605339 C2

FIELD: medicine; pharmaceuticals.

SUBSTANCE: invention relates to medicine and pharmaceutical industry and represents therapeutic agent, based on amantadine sulphate, for reduction of glutamate-induced apoptosis and inhibition of NMDA-receptors for treating nervous system disorders, effects of craniocereberal injury and ischemic and hemorrhagic stroke, characterized by that it contains therapeutically effective amount of amantadine sulphate and cytidine 5'-diphosphocholine as active substance, as well as at least one auxiliary substance, selected from group consisting of stabilizers, prolongators, buffering additive solvents, fillers, preserving agents, ingredients are taken in certain ratio, wt%.

EFFECT: invention provides extending of range of products for reduction of glutamate-induced apoptosis and inhibition of NMDA-receptors for treating disorders of nervous system, effects of craniocereberal injury and ischemic and hemorrhagic stroke, increase of clinical effectiveness, stability at room temperature, long storage life, at least 3 years.

4 cl, 3 ex, 3 tbl

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RU 2 605 339 C2

Authors

Khoroshilova Galina Vladimirovna

Koverda Mikhail Nikolaevich

Zemljanukhina Ekaterina Sergeevna

Dates

2016-12-20Published

2013-07-23Filed