FIELD: chemistry.
SUBSTANCE: invention relates to a process of preparation of aroyl pyruvic acid N-arylamides of the general formula I-III
,
wherein
.
The process of N-arylamides of aroyl pyruvic acids is carried out by boiling the arylamines with methyl esters of aroylpyruvic acids in glacial acetic acid for 15-20 minutes in the presence of anhydrous sodium acetate.
EFFECT: preparation of N-arylamides of aroyl pyruvic acids in high yield, in the absence of dry solvents and toxic reagents.
3 ex
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Authors
Dates
2017-07-03—Published
2014-12-01—Filed