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(19)

(11)

2 627 269

(13)

(51)

IPC

C07D498/04(2006-01-01)

A61K31/519(2006-01-01)

A61P3/04(2006-01-01)

A61P9/00(2006-01-01)

A61P11/00(2006-01-01)

A61P33/00(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2014134640, 2013-01-25

(24)

Start date

2013-01-25

(22)

Actual filing date

2013-01-25

(45)

Published

2017-08-04

(72)

Inventor

Bron AlenKrespen OliveForishe IanMarsinyak ZhilberMyuze NikolyaNikole ErikPaskal SesilVive BertranVivyani Fabris

(73)

Holder

Sanofi

BICYCLIC HETEROCYCLIC DERIVATIVES, THEIR PRODUCTION AND APPLICATION Russian patent published in 2017 - IPC C07D498/04 A61K31/519 A61P3/04 A61P9/00 A61P11/00 A61P33/00 A61P35/00

Abstract RU 2627269 C2

FIELD: pharmacology.

SUBSTANCE: invention relates to compounds of general formula (I) , as well as to a method for their preparation, pharmaceutical compositions based thereon, and their application.

EFFECT: new compounds have been obtained that can be used to treat or prevent pathology for which it is necessary to inhibit the mTOR kinase.

20 cl, 4 tbl, 30 ex

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RU 2 627 269 C2

Authors

Bron Alen

Krespen Olive

Forishe Ian

Marsinyak Zhilber

Myuze Nikolya

Nikole Erik

Paskal Sesil

Vive Bertran

Vivyani Fabris

Dates

2017-08-04—Published

2013-01-25—Filed