NOVEL COMPOUNDS THAT ARE ERK INHIBITORS Russian patent published in 2018 - IPC C07D471/04 C07D471/16 C07D498/16 C07D498/18 C07D513/04 C07D519/00 A61K31/437 A61K31/4375 A61K31/496 A61K31/5377 A61K31/553 A61K45/06 A61P35/00 

Abstract RU 2660429 C2

FIELD: chemistry.

SUBSTANCE: invention relates to compounds of formula (1) in which the radicals and symbols have the meanings indicated in the claims and to pharmaceutically acceptable salts thereof. Compounds of formula (1) are ERK inhibitors.

.

EFFECT: invention also relates to a pharmaceutical composition comprising and to methods for treating malignant neoplasms using a compound of formula (1).

16 cl, 6 tbl, 458 ex

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RU 2 660 429 C2

Authors

Uilson Kevin Dzh.

Uitter Devid Dzh.

Silipkhaivankh Pkhieng

Lipford Ketrin

Sloman Devid

Falkone Deniell

O'Bojl Brendan

Mansur Umar Faruk

Lim Chzhongvon

Metot Dzhoi L.

Bojs Kristofer

Chen Lej

Deniels Mettyu Kh.

Fevrier Salem

Khuan Syankhaj

Kurukulasuriya Ravi

Tun Lin

Chzhou Vej

Kozlovski Dzhozef

Maletik Milana M.

Shinkre Bidkhan A.

Tkhataj Dzhayantkh Tkhiruvellore

Bakshi Raman Kumar

Karunakaran Ganesh Babu

Dates

2018-07-06Published

2013-09-26Filed