[1,2,4] TRIAZOLOPIRIDINES AND THEIR APPLICATION AS INHIBITORS OF PHOSPHODIESTERASE Russian patent published in 2017 - IPC C07D471/04 A61K31/437 A61P11/06 A61P17/00 

Abstract RU 2630699 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a compound of general formula (I)

in which R is a branched butyl. The invention also relates to a pharmaceutical composition having a phosphodiesterase inhibitory activity, to the use of a compound for the preparation of a pharmaceutical composition, and to a method of treating or reducing the intensity of a disease, disorder or condition susceptible to a PDE4 inhibitory activity.

EFFECT: new compound of general formula I, having a phosphodiesterase inhibitory activity, was obtained.

10 cl, 4 ex

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RU 2 630 699 C2

Authors

Nilsen Simon Feldbek

Larsen Jens Khristian Khojlann

Dates

2017-09-12Published

2012-12-19Filed