NEW METHOD OF SYNTHESIS OF TETRAHYDROPYRASIN[2,3-C]PYRIDAZINE DERIVATIVES Russian patent published in 2017 - IPC C07D487/04 A61K31/5025 A61P35/00 

Abstract RU 2631430 C1

FIELD: pharmacology.

SUBSTANCE: invention relates to a method for synthesis of tetrahydropyrazino[2,3-c]pyridazine derivatives of the formula , which can be used for manufacture of medicaments for treatment of oncological, chronic inflammatory and other diseases.

EFFECT: new synthesis method allows to obtain compounds of general formula 1 possessing an increased degree of purity.

7 cl, 6 dwg, 5 ex

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RU 2 631 430 C1

Authors

Titov Ilya Yurevich

Stroganov Oleg Valentinovich

Chilov Germes Grigorevich

Strojlov Viktor Sergeevich

Novikov Fedor Nikolaevich

Dates

2017-09-22Published

2016-10-26Filed