CYCLOALKANE DERIVATIVE Russian patent published in 2017 - IPC C07D285/08 C07D401/12 C07D403/12 C07D417/12 A61K31/427 A61K31/433 A61K31/506 A61P25/00 A61P29/00 

Abstract RU 2635354 C2

FIELD: pharmacology.

SUBSTANCE: invention provides a compound represented by the formula , or a pharmacologically acceptable salt thereof, where Ar1 and Ar2: a heteroaryl group or an aryl group; R1, R2 and R3: a hydrogen atom, a halogen atom, a C1-C6 alkyl group, a halogenated C1-C6 alkyl group or a cyano group; R4 and R5: a hydrogen atom, a halogen atom, a C1-C6 alkyl group, a hydroxyl group or a C1-C6 alkoxy group; N: an integer between 1 and 3; and the heteroaryl group or aryl group optionally contains one or two groups, independently selected from a halogen atom, a C1-C6 alkyl group, an amino group, and when a heteroaryl group or aryl group contains two such groups, the two groups are the same or different.

EFFECT: increased efficiency of treatment.

33 cl, 5 dwg, 8 tbl, 179 ex

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RU 2 635 354 C2

Authors

Sinozuka Tsuesi

Kobayasi Khiroyuki

Suzuki Sayaka

Tanaka Kesuke

Kimoto Khiroko

Domon Yuki

Dates

2017-11-13Published

2013-02-08Filed