COMPOSITION FOR ASTHMA PREVENTION OR TREATMENT CONTAINING MONOACETHYLDIACYL GLYCERINE COMPOUND AS ACTIVE INGREDIENT Russian patent published in 2017 - IPC A61K31/22 A61K47/00 A61P11/06 

Abstract RU 2636615 C2

FIELD: pharmacology.

SUBSTANCE: monoacetyl diacylglycerin according to the invention is a natural substance isolated from deer antlers. The monoacetyl diacylglycerols of the invention inhibit the expression of interleukin-4 (IL-4) in mouse T-cell lymphoma cells (EL-4), reduce airway hyperreactivity in experimental induced asthma in animals, and inhibit inflammatory cells penetration into the bronchial tree. In addition, the compounds of the invention reduce the immunoglobulin E (IgE) content in the blood serum and in the fluid obtained from bronchoalveolar lavage; have a pronounced effect of suppressing the expression of cytokines produced by Th2 cells (IL-4, IL-5 and IL-13) in the lungs, and have no side effects, are not toxic, and have an effective therapeutic effect.

EFFECT: asthma prevention or treatment.

9 cl, 7 dwg, 7 tbl, 8 ex

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RU 2 636 615 C2

Authors

O Sej-Ryan

An Kyun Sop

Li Su Ui

Sin In Sik

Sin Na-Ne

Li Te-Sok

Kan Chonko

Chon Yun-Sik

Khan En-Khe

Son Ki En

Dates

2017-11-24Published

2014-08-19Filed