FIELD: pharmacology.
SUBSTANCE: monoacetyl diacylglycerin according to the invention is a natural substance isolated from deer antlers. The monoacetyl diacylglycerols of the invention inhibit the expression of interleukin-4 (IL-4) in mouse T-cell lymphoma cells (EL-4), reduce airway hyperreactivity in experimental induced asthma in animals, and inhibit inflammatory cells penetration into the bronchial tree. In addition, the compounds of the invention reduce the immunoglobulin E (IgE) content in the blood serum and in the fluid obtained from bronchoalveolar lavage; have a pronounced effect of suppressing the expression of cytokines produced by Th2 cells (IL-4, IL-5 and IL-13) in the lungs, and have no side effects, are not toxic, and have an effective therapeutic effect.
EFFECT: asthma prevention or treatment.
9 cl, 7 dwg, 7 tbl, 8 ex
Title |
Year |
Author |
Number |
COMPOSITION FOR PREVENTION OR TREATMENT OF CHRONIC OBSTRUCTIVE PULMONARY DISEASES CONTAINING MONOACETHYLDIGLYCEROL COMPOUNDS AS ACTIVE INGREDIENT |
2014 |
- O Sej-Ryan
- An Kyun Sop
- Li Su Ui
- Sin In Sik
- Kvon Ok-Kyun
- Kim Syn Khyun
- Chun Chan Mi
- Li Te-Sok
- Khan En-Khe
- Son Ki En
- Kan Chonko
- Kim Khe Kyun
|
RU2642631C2 |
COMPOSITION FOR DETECTION OF CANCER BLOOD DISEASES OR METASTASIS OF CANCER CONTAINING ACTIVE INGREDIENT MONOACETHYL DIGLYCERIDE COMPOUND |
2014 |
- Kim Che Khva
- O Sej Ryan
- An Kyun Sop
- Kan Kho Pum
- Sin Che Min
- Ko Yun Yn
- Li Te Sok
- Kim Men Khvan
- Kan Chon Ko
- Khan En-Khe
- Son Ki-Yun
|
RU2632098C2 |
COMPOSITIONS CONTAINING MONOACETYLDIACYLGLYCERIDE AS AN ACTIVE INGREDIENT FOR PREVENTING OR TREATING RHEUMATOID ARTHRITIS |
2014 |
- Kim Che Khva
- O Sej Ryan
- An Kyun Sop
- Kan Kho Pum
- Pek Pom Su
- Li Te-Sok
- Kan Chon Ko
- Chon Yun-Sik
- Khan En-Khe
- Son Ki En
|
RU2646823C2 |
COMPOSITION FOR ATOPIC ECZEMA PREVENTION OR TREATMENT CONTAINING MONOACETYLDIACYL GLYCERINE COMPOUND AS ACTIVE INGREDIENT |
2014 |
- Kim Che Khva
- O Sej-Ryan
- An Kyun Sop
- Kan Kho Pum
- Yu Che Mine
- Li Te-Sok
- Kan Chonko
- Kim Khe Kyun
- Yuk Chin Su
- Khan En-Khe
- Son Ki En
|
RU2640503C2 |
NEW COMPOUND ISOLATED FROM PSEUDOLYSIMACHION ROTUNDUM VAR. SUBINTEGRUM, WITH A HIGH CONTENT OF ACTIVE INGREDIENT, COMPOSITION CONTAINING SAID COMPOUND FOR PREVENTING OR TREATING ALLERGIC DISEASE, INFLAMMATORY DISEASE, ASTHMA OR CHRONIC OBSTRUCTIVE PULMONARY DISEASE AND USE THEREOF |
2015 |
- Li Ennam
- Yu Chi-Sok
- Sin Te-Khi
- Yu Pen-Khvan
- O Si-Yan
- An Ken-Sop
- Li Khen-Ke
- Li Su Uj
- Son Khek-Khvan
- Sin In-Sik
- Yu Khen Von
|
RU2685732C2 |
METHODS OF TREATING LEUKOPENIA AND THROMBOCYTOPENIA |
2015 |
- Khan En-Khe
- Chon Sekho
- Son Ki-Yun
- Kim Men-Khvan
- Kim Che Khva
|
RU2702122C2 |
IMMUNOMODULATORY AGENT, CANCER AGENT AND HEALTHY FOOD CONTAINING MONOACETYLDIACYLGLYCERIN DERIVATIVES |
2005 |
|
RU2341257C2 |
COMPOSITIONS FOR PREVENTING OR TREATING ACUTE RADIATION SICKNESS |
2018 |
- Sohn, Ki Young
- Yoon, Sun Young
|
RU2841262C2 |
LACTOBACILLUS CRISPATUS KBL693 STRAIN AND ITS APPLICATION |
2019 |
- Ko, Vu Ri
- Li, Dzhun Chkhul
- Nam, Te Vuk
- Ko, Kvan Pe
- Yu, Khen Dzhu
- Yun, So En
- Son, Sok Chkhon
|
RU2791561C2 |
FOOD BUTYRATE FOR TREATMENT OR PREVENTION OF ALLERGIC DISORDER |
2019 |
- Blanchard, Carine
- Bourdeau, Tristan
- Destaillats, Frederic
- Forbes-Blom, Elizabeth
- Nutten, Sophie
- Oertling, Heiko
- Patin, Amaury
|
RU2809650C2 |