CHEMICAL METHOD Russian patent published in 2018 - IPC C07D211/14 

Abstract RU 2644160 C2

FIELD: chemistry.

SUBSTANCE: invention relates to the method of producing a compound of the formula , where R1 is C1-6alkyl, aryl, or benzyl, and Y is a leaving group, which includes: a) the interaction of the compound of the formula with 2-chloroethanol in the presence of a suitable base; and b) the conversion of the product obtained in step (a) into the compound of the formula (V) using a reagent selected from the group consisting of thionyl chloride, sulphonylchloride such as sulphonylchlorides, sulfonyl anhydrides, and halides of phosphorus.

EFFECT: improved method.

7 cl, 8 dwg, 1 tbl, 10 ex

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RU 2 644 160 C2

Authors

Hossner Frank

Strachan John Bryce

Dates

2018-02-08Published

2013-08-14Filed