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2 650 877

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IPC

C07D487/04(2006-01-01)

A61K31/4184(2006-01-01)

A61K31/4188(2006-01-01)

A61P3/10(2006-01-01)

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Application

2017137204, 2017-10-23

(24)

Start date

2017-10-23

(22)

Actual filing date

2017-10-23

(45)

Published

2018-04-18

(72)

Inventor

Zhukovskaya Olga NikolaevnaSpasov Aleksandr AlekseevichBabkov Denis AleksandrovichMorkovnik Anatolij Savelevich

(73)

Holder

Federalnoe Gosudarstvennoe Avtonomnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniya Federalnyj Universitet"Federalnoe Gosudarstvennoe Byudzhetnoe Obrazovatelnoe Uchrezhdenie Vysshego Obrazovaniya Gosudarstvennyj Meditsinskij Universitet" Ministerstva Zdravookhraneniya Rossijskoj Federatsii

HYDROBROMID 4'-(2,3-DIGIDRO-9H-IMIDAZO[1,2-A]BENZIMIDAZOLE-9-YL-METHYL)BIPHENYL-2-CARBONITRIL EXHIBITING THE PROPERTIES OF THE ACTIVATOR OF AMP-ACTIVATED PROTEINKINASE (AMPA) Russian patent published in 2018 - IPC C07D487/04 A61K31/4184 A61K31/4188 A61P3/10

Abstract RU 2650877 C1

FIELD: chemistry.

SUBSTANCE: invention relates to the field of organic chemistry, namely to hydrobromide 4'- (2,3-dihydro-9H-imidazo[1,2-a]benzimidazol-9-yl-methyl)biphenyl-2-carbonitrile of formula I.

EFFECT: new compound is obtained in the series of derivatives 2,3-dihydroimidazo[1,2-a]benzimidazole, exhibiting the properties of the AMPK activator.

1 cl, 1 dwg, 1 tbl, 2 ex

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RU 2 650 877 C1

Authors

Zhukovskaya Olga Nikolaevna

Spasov Aleksandr Alekseevich

Babkov Denis Aleksandrovich

Morkovnik Anatolij Savelevich

Dates

2018-04-18—Published

2017-10-23—Filed