Show metadata Hide metadata

(19)

(11)

2 654 851

(13)

(51)

IPC

C07C315/04(2006-01-01)

A61K31/255(2006-01-01)

A61P17/00(2006-01-01)

(21) (22)

Application

2015139778, 2015-09-18

(24)

Start date

2015-09-18

(22)

Actual filing date

2015-09-18

(45)

Published

2018-05-23

(72)

Inventor

Akhmetova Vnira RakhimovnaAkhmadiev Nail SalavatovichGalimzyanova Nailya FauatovnaIbragimov Askhat GabdrakhmanovichDzhemilev Usein Memetovich

(73)

Holder

Federalnoe Gosudarstvennoe Byudzhetnoe Nauchnoe Uchrezhdenie Ufimskij Federalnyj Issledovatelskij Tsentr Rossijskoj Akademii Nauk Ran)

METHOD FOR PRODUCING 3-SULFANYLMETHYL-DERIVATIVES OF 2,4-PENTANDIONE THAT HAS ANTI-FUNGAL ACTIVITY IN RESPECT OF TRICHOPHYTON TERRESTERE Russian patent published in 2018 - IPC C07C315/04 A61K31/255 A61P17/00

Abstract RU 2654851 C2

FIELD: pharmacology.

SUBSTANCE: interaction of the mixture of formaldehyde and tert-butylthiol (tiophenol) with 2,4-pentandione involving promoter BuONa in molar ratio of formaldehyde: tert-butylthiol (tiophenol): 2,4-pentadione: BuONa=1:1:1:1 in a mixture of solvents CHCl₃-C₂H₅OH (1:1, vol.), at room temperature (~20°C) and atmospheric pressure for 5-7 h.

EFFECT: anti-fungal activity against pathogenic Trichophyton dermatomycetes.

2 cl, 2 tbl, 7 ex

Similar patents RU2654851C2

Title	Year	Author	Number
PRODUCTION METHOD FOR 3-[(PHENYLSULFENYL)METHYL]PENTANE-2,4-DIONE SHOWING A FUNGICIDAL ACTIVITY	2015	Akhmetova Vnira Rakhimovna Akhmadiev Nail Salavatovich Galimzyanova Nailya Fauatovna Ibragimov Askhat Gabdrakhmanovich Dzhemilev Usein Memetovich	RU2615155C2
METHOD OF PRODUCING α-[(PENTANE-2,4-DION-3-YL)METHOXY]-ω-[(PENTANE-2,4-DION-3-YL)METHYLSULPHANYL] ALKANES	2014	Akhmadiev Nail Salavatovich Akhmetova Vnira Rakhimovna Kunakova Rajkhana Valiulovna Ibragimov Askhat Gabdrakhmanovich Dzhemilev Usein Memetovich	RU2605450C2
METHOD FOR PRODUCING 1,2(1,5)-{BIS[ALKYL-(2-CYANO-3-SULPHANYL)PROPANOATE]}ETHANE(SULPHANE-3-YLPENTANES)	2021	Akhmadiev Nail Salavatovich Sharafutdinova Ruzalina Radikovna Ibragimov Askhat Gabdrakhmanovich Dzhemilev Usein Memetovich	RU2780151C1
2-PHENYLTHIOMETHYL SUBSTITUTED 1,3-DIKETONES AND DIMETHYLMALONATE - AGENT HAVING FUNGICIDAL ACTIVITY	2015	Galimzyanova Nailya Fauatovna Akhmadiev Nail Salavatovich Akhmetova Vnira Rakhimovna Zajnullin Radik Anvarovich Kunakova Rajkhana Valiullovna	RU2616603C2
METHOD OF OBTAINING α, ω-{ BIS[(PENTAN-2,4-DION-3-YL)METHYLSULPHANYL]}-ALKANES	2012	Dzhemilev Usein Memetovich Akhmetova Vnira Rakhimovna Akhmadiev Nail' Salavatovich Sufijarova Roza Shajkhal'Nurovna Ibragimov Askhat Gabdrakhmanovich	RU2529514C2
METHOD OF PRODUCING 1,8-{BIS[(PENT-2,4-DION-3-YL)METHYLSULPHANYL]}-3,6-DIOXAOCTANE AND 4,4'-{BIS[(PENT-2,4-DION-3-YL)METHYLSULPHANYL]}-DIPHENYL OXIDE	2012	Dzhemilev Usein Memetovich Akhmetova Vnira Rakhimovna Akhmediev Nail' Salavatovich Veklov Vitalij Aleksandrovich Gabdrakhmanova Rushana Floridovna Ibragimov Askhat Gabdrakhmanovich	RU2529512C2
METHOD OF OBTAINING N,N-DIMETHYL-N-[(ALKYLSULFANYL)METHYL]AMINES	2010	Dzhemilev Usein Memetovich Khajrullina Regina Radievna Akmanov Bajras Faritovich Ibragimov Askhat Gabdrakhmanovich Akhmetova Vnira Rakhimovna Kunakova Rajkhana Valiullovna	RU2466985C2
METHOD OF OBTAINING N,N,N,N-TETRASUBSTITUTED DI[4-(AMINOMETHYLSULFANYL)]PHENYL ETHERS	2011	Dzhemilev Usein Memetovich Khajrullina Regina Radievna Akmanov Bajras Faritovich Ibragimov Askhat Gabdrakhmanovich Kunakova Rajkhana Valiullovna Popod'Ko Natal'Ja Romanovna	RU2466987C1
METHOD OF PRODUCING 2-[(ALKYL(PHENYL)SULFANYL)METHYL]BENZAMIDES	2022	Khairullina Regina Radievna Tiumkina Tatiana Viktorovna	RU2788745C1
STEROIDS, A METHOD OF SYNTHESIS OF STEROIDS, A METHOD OF SYNTHESIS OF 16-METHYLENESTEROIDS, COMPOUNDS	1992	Zhan Buavehn[Fr] Kristin Shove[Fr] Samir Zard[Lb]	RU2099346C1

RU 2 654 851 C2

Authors

Akhmetova Vnira Rakhimovna

Akhmadiev Nail Salavatovich

Galimzyanova Nailya Fauatovna

Ibragimov Askhat Gabdrakhmanovich

Dzhemilev Usein Memetovich

Dates

2018-05-23—Published

2015-09-18—Filed