PYRAZINO[1,2-A]INDOLE COMPOUNDS, PREPARATION AND USE THEREOF IN MEDICAMENTS Russian patent published in 2018 - IPC C07D487/04 A61K31/4985 A61P29/00 

Abstract RU 2660417 C2

FIELD: chemistry.

SUBSTANCE: invention relates to compounds of general formula (I), as well as to pharmaceutically acceptable salts, enantiomers, diastereomer or racemates thereof. .

EFFECT: technical result: novel compounds having sigma receptor activity, that are useful for the treatment and/or prophylaxis of sigma mediated diseases or conditions.

8 cl, 2 tbl, 3 ex

Similar patents RU2660417C2

Title Year Author Number
BIOMARKER ANALYSIS FOR DETECTING OR MEASURING TOR-KINASE ACTIVITY INHIBITION 2011
  • Vong Lilli
  • Syuj Shujchan
  • Din Tszyan-Khua
RU2587040C2
USE OF SIGMA LIGANDS WITH INDUCED OPIOIDS HYPERALGESIA 2011
  • Vela Ernandes Khose Migel
  • Samanilo-Kastanedo Daniel
  • Puig Rera De Konias Margarita
RU2589899C2
USE OF SIGMA LIGANDS FROM PAIN IN BONE CANCER 2011
  • Samanilo-Kastanedo Daniel
  • Vela-Ernandes Khose Migel
  • Plata-Salaman Karlos
RU2585095C2
SIGMA-LIGANDS FOR APPLICATION IN PREVENTION AND/OR TREATMENT OF POSTOPERATIVE PAIN 2011
  • Vela Ehrnandes Khose Migel'
  • Samanil'O-Kastanedo Daniehl'
  • Puig-R'Era De Konias Margarita
RU2569055C2
METHODS OF OBTAINING AND PURIFICATION OF HETEROARYL COMPOUNDS 2010
  • Kharris Roj L.
  • Sapienza Dzhon
  • Shevlin Graziehlla
  • Papa Patrik
  • Li Brenden Dzhingsi
  • Pakard Garrik
  • Chzhao Tszintszin
  • Dzhokil Patrik Ehntoni
  • Mortensen Debora
  • Riggs Dzhennifer
  • Gamboa Khuan Antonio
  • Bosham Mehri Dzhordzh
  • Krejlejn Mehtt'Ju Majkl
  • Kotare Mokhit Atul
  • Perren-Ninkovich Sofi
  • Paj Filip
  • Leong Uill'Jam Vehj-Khva
  • Ehl'Sner Jan
  • Choudkhuri Anusuja
RU2557242C2
mTOR KINASE INHIBITORS FOR ONCOLOGICAL INDICATIONS AND DISEASES METABOLICALLY BOUND TO mTOR/PI3K/AKT 2009
  • Ehl'Sner Jan
  • Kharris Roj L.
  • Li Brehnden
  • Mortensen Debora
  • Pakard Garrik
  • Papa Patrik
  • Perren-Ninkovich Sofi
  • Riggs Dzhennifer
  • Sankar Sabita
  • Sapienza Dzhon
  • Shevlin Graziehlla
  • Terani Lida
  • Sjuj Vehjmin
  • Chzhao Tszintszin
  • Parnes Dzhejson
  • Madakamutil Lui
  • Fults Kimberli
  • Narla Rama K.
RU2546658C2
MTOR KINASE INHIBITORS FOR ONCOLOGIC INDICATIONS AND DISEASES ASSOCIATED WITH MTOR/PI3K/AKT BY METABOLISM 2009
  • Elsner Yan
  • Kharris Roj L.
  • Li Brenden
  • Mortensen Debora
  • Pakard Garrik
  • Papa Patrik
  • Perren-Ninkovich Sofi
  • Riggs Dzhennifer
  • Sankar Sabita
  • Sapienza Dzhon
  • Shevlin Graziella
  • Terani Lida
  • Syuj Vejmin
  • Chzhao Tszintszin
  • Parnes Dzhejson
  • Madakamutil Lui
  • Fults Kimberli
  • Narla Rama K.
RU2692796C2
IDENTIFICATION OF LKB1 MUTATION AS PROGNOSTIC BIOMARKER OF SENSITIVITY TO TOR-KINASE INHIBITORS 2011
  • Sankar Sabita
  • Chopra Radzhesh
  • Sjuj Vehjmin
  • Nin Jujkhun
  • Sju Shujchan'
RU2565034C2
ESTROGEN RECEPTOR MODULATORS 2017
  • Khuan Piter Tsinkhua
  • Sli Debora Khelen
  • Khegde Saji Gadzhanan
  • Khopkins Chad Deniel
  • Banker Kevin Duejn
  • Pinchman Dzhozef Robert
  • Sit Rakesh Kumar
RU2738646C2
SIGMA-RECEPTOR INHIBITORS 2005
  • Laggner Kristian
  • Kuberes-Altisent Marija Rosa
  • Kholents Jorg
  • Berrokal'-Romero Khuana Marija
  • Kontikhoch-L'Obet Marija Montserrat
RU2417987C2

RU 2 660 417 C2

Authors

Merse-Vidal Ramon

Dias Fernandes Khose Luis

Almansa Rosales Karmen

Dates

2018-07-06Published

2014-04-22Filed