PYRAZOLE COMPOUNDS AS MODULATORS OF FSHR AND USES THEREOF Russian patent published in 2018 - IPC C07D491/52 A61P15/08 A61K31/4162 

Abstract RU 2663898 C2

FIELD: chemistry.

SUBSTANCE: invention relates to a compound of formula I,

or a pharmaceutically acceptable salt thereof, also to a pharmaceutical composition, methods of treatment and modulation, due to the effect on the receptor of follicle-stimulating hormone.

EFFECT: compounds of this invention, and pharmaceutically acceptable compositions thereof, are effective as modulators of FSHR.

19 cl, 50 ex

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RU 2 663 898 C2

Authors

Yuj Genri

Donnelli Merien

Ngujen Ngan

Tszyan Syujlyan

Dates

2018-08-13Published

2014-06-24Filed