HETEROARYL COMPOUNDS AS TKB INHIBITORS AND USE THEREOF Russian patent published in 2021 - IPC C07D471/04 C07D519/00 A61K31/437 A61K31/553 A61P29/00 A61P37/00 

Abstract RU 2742122 C2

FIELD: pharmaceuticals.

SUBSTANCE: present invention relates to an imidazopyridine compound of formula I and pharmaceutically acceptable salts thereof, the structural formulas of which are given in the claim.

I

EFFECT: imidazopyridine compounds according to the invention are intended as Bruton's tyrosine kinase inhibitor (BTK).

3 cl, 5 tbl, 190 ex

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RU 2 742 122 C2

Authors

Gaillard, Pascale

Seenisamy, Jeyaprakashnarayanan

Gardberg, Anna

Johnson, Theresa L.

Sherer, Brian A.

Goutopoulos, Andreas

Won, Annie Cho

Jones, Reinaldo

Neagu, Constantin

Qiu, Hui

Caldwell, Richard D.

Potnick, Justin

Liu-Bujalski, Lesley

Dates

2021-02-02Published

2015-10-06Filed