PYRAZOLE-AMIDE COMPOUND AND MEDICINAL USES THEREFOR Russian patent published in 2018 - IPC C07D231/12 A61K31/415 A61P3/04 A61P3/10 A61P9/04 A61P9/10 A61P11/00 A61P13/12 A61P25/00 A61P27/02 A61P27/12 A61P43/00 

Abstract RU 2664532 C2

FIELD: medicine; pharmaceuticals.

SUBSTANCE: invention relates to a compound of the formula [I] wherein n is 1 or 2, or to its corresponding pharmaceutically acceptable salts. Invention also relates to compounds represented by formulas [II], [IIh] and [III]. Pharmaceutical use of these compounds is also described.

EFFECT: these compounds are an inhibitor of PDHK (PDHK1 and / or PDHK2).

15 cl, 2 dwg, 6 tbl, 2 ex

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RU 2 664 532 C2

Authors

Motomura Takakhisa

Semi Gakudzun

Dates

2018-08-20Published

2014-03-14Filed