CRYSTAL AND SALT FORMS OF PPAR AGONIST COMPOUNDS Russian patent published in 2021 - IPC C07D233/64 C07D401/04 A61K31/4174 A61K31/4439 A61P35/00 

Abstract RU 2759724 C2

FIELD: organic chemistry.

SUBSTANCE: invention relates to the field of organic chemistry, namely to hemisulfate salt of a compound of the formula (I) and megluminous salt or hydrate of megluminous salt of a compound of the formula (II). The invention also relates to crystal forms of the specified salts, a pharmaceutical composition based on the specified compounds, and a method for treating a PPARδ-related disease or condition in a subject that provides for the injection of therapeutically effective amount of the specified compounds or a pharmaceutical composition to a subject who needs it.

EFFECT: new compounds with the capability of enhancing PPARδ activity are obtained.

19 cl, 2 dwg, 6 tbl, 14 ex

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RU 2 759 724 C2

Authors

Lagu, Bkharat

Tshaska, Skott

Dates

2021-11-17Published

2017-10-05Filed