5-AZAINDAZOLE COMPOUNDS AND METHODS FOR USE THEREOF Russian patent published in 2018 - IPC C07D471/04 C07D471/10 C07D487/10 A61K31/437 A61P35/00 A61P29/00 A61P9/00 A61P37/00 

Abstract RU 2665462 C2

FIELD: chemistry.

SUBSTANCE: invention relates to particular compounds which are derivatives of 5-azaindazole, which are indicated in the claims. Said compounds are useful for inhibiting Pim kinase and for treating diseases such as cancer mediated by Pim kinase.

EFFECT: disclosed are methods of using compounds of formula (I) in vitro, in situ and in vivo to diagnose, prevent or treat similar diseases in mammalian cells or related pathological conditions.

6 cl, 4 tbl, 188 ex

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RU 2 665 462 C2

Authors

Deu Stiven

Khu Khuejyun

Kolesnikov Aleksandr

Tsui Viki Kh.

Van Syaotszin

Dates

2018-08-30Published

2013-06-26Filed