FIELD: chemical-pharmaceutical industry.
SUBSTANCE: invention relates to a novel chromon oxime derivative of formula (I), also relates to pharmaceutical compositions containing said compound, and to their use in the treatment or prevention of conditions associated with altered glutamatergic signaling and/or function, or conditions that can be influenced, changing the level of glutamate or signal transmission, in particular Parkinson's disease.
.
EFFECT: technical result: new compound of formula (I) is obtained which is a modulator of brain permeability mGluRs of the nervous system and, in addition, provides an advantageous high permeability of the brain after oral administration.
14 cl, 10 dwg, 3 ex, 3 tbl
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Authors
Dates
2018-11-16—Published
2015-08-27—Filed