NITROIMIDAZOLE DERIVATIVE AGAINST PULMONARY TUBERCULOSIS Russian patent published in 2018 - IPC C07D519/00 C07D498/04 A61K31/519 A61P31/06

Abstract RU 2675622 C1

FIELD: medicine; pharmaceuticals.

SUBSTANCE: invention relates to new derivatives of nitroimidazole of formula (I), as well as to a pharmaceutical composition based on them and use for the manufacture of a medicament for the treatment of diseases caused by Mycobacterium tuberculosis. .

EFFECT: technical result: new compounds with inhibitory activity against Mycobacterium tuberculosis, which, in addition, have high solubility and permeability.

11 cl, 1 tbl

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RU 2 675 622 C1

Authors

Luo, Wei

Ding, Charles Z.

Huang, Zhigang

Chen, Shuhui

Dates

2018-12-21—Published

2016-01-28—Filed