FUNCTIONALISED BENZOPYRAN COMPOUNDS AND USE THEREOF Russian patent published in 2019 - IPC C07D311/16 C07D311/58 C07D407/04 A61K31/353 A61P35/00 

Abstract RU 2676766 C2

FIELD: chemistry.

SUBSTANCE: invention relates to the compound of general formula (I)

where R1 is selected from the group consisting of: H and C1-C6 alkyl, R2 represents OH, R3 is selected from the group consisting of: H, C1-C6 alkyl and halogen, radicals from R10 to R12 are independently selected from the group consisting of: OH, C1-C6 alkyl, C1-C6 alkoxy and halogen, R13 is selected from the group consisting of: OH, C1-C6 alkoxy, NH2, NHMe, NHEt, N(Me)2 and N(Et)2, R14 and R15 are independently selected from the group consisting of: H, C1-C6 alkyl and halogen, or R13 and one of R14 and R15 form following structure: Also, the invention relates to a method for producing said compound and a pharmaceutical composition based thereon.

EFFECT: new compounds and a pharmaceutical composition based on them have been obtained that can be used in medicine for treatment of cancer.

52 cl, 12 dwg, 6 tbl, 6 ex

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RU 2 676 766 C2

Authors

Khiton Endryu

Braun Devid

Kelli Grekhem

Dates

2019-01-11Published

2015-02-05Filed