AMORPHOUS FORM OF THIOCOLCHICINE COMPOUND Russian patent published in 2019 - IPC C07C319/28 C07C323/44 A61K31/17 

Abstract RU 2684925 C2

FIELD: chemical-pharmaceutical industry.

SUBSTANCE: invention relates to an amorphous form of a compound of formula (I) having an XRPD (X-ray powder diffraction) pattern, which is shown in Fig. 1. Invention also relates to a method for preparing said amorphous form and pharmaceutical compositions containing said composition.

.

EFFECT: said form has improved stability compared to crystalline forms and can find application, in particular, in treating solid tumors.

8 cl, 8 dwg, 3 ex

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RU 2 684 925 C2

Authors

Cabri Walter

Peterlongo Federico

Ciceri Daniele

Gambini Andrea

Dates

2019-04-16Published

2015-03-26Filed