FIELD: medicine.
SUBSTANCE: invention is related to a compound represented by the formula
and its pharmaceutically acceptable salt. The invention is also related to a complex and a co-crystal containing said compound and fumaric acid in a 1:1 molar ratio, with an X-ray powder diffraction pattern having peaks at diffraction angles (2θ): 9.5±0.2°, 10.9±0.2°, 18.6±0.2°, 23.5±0.2° and 24.6±0.2°.
EFFECT: obtaining a new compound, as well as a complex and a co-crystal based on it with fumaric acid, which can be used in medicine for the treatment and/or prevention of a disease associated with coronavirus 3CL proteases.
12 cl, 13 dwg, 8 tbl, 6 ex
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Authors
Dates
2023-10-25—Published
2022-02-17—Filed