4-AMINO-1-{2-[3-METHYL-5-(BENZENESULFONYLOXY]PHENOXY]ETHYL}-PYRIDIUM CHLORIDE SUBSTANCE, HAVING THE BIOLOGICALLY ACTIVE AGENT PROPERTIES, INFLUENCING THE MAMMALS BLOOD COAGULABILITY NATURALLY RUNNING PROCESSES, ANTICOAGULANT ON ITS BASIS AND ITS OBTAINING METHOD BY CHEMICAL SYNTHESIS Russian patent published in 2019 - IPC C07D213/64 A61K31/44 A61P7/02 

Abstract RU 2685261 C1

FIELD: chemistry.

SUBSTANCE: group of inventions relates to the 4-amino-1-{2-[3-methyl-5-(benzenesulfonyloxy]phenoxy]ethyl}-pyridium chloride, having the structural formula

,

which is the thrombin direct inhibitor, as well as to its production and application method.

EFFECT: ensuring the biologically active substance, the thrombin inhibitor, oral administration possibility, and at that preserving its specific pharmacological activity as the anticoagulant.

4 cl, 1 dwg, 5 tbl

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RU 2 685 261 C1

Authors

Plotnikov Mark Borisovich

Zavarzin Igor Viktorovich

Nazarov Andrej Konstantinovich

Kuznetsov Yurij Vladimirovich

Kachanov Oleg Yurevich

Dates

2019-04-17Published

2018-04-05Filed