SUBSTITUTED IMIDAZOPYRIDINES AS HDM2 INHIBITORS Russian patent published in 2019 - IPC C07D471/04 A61K31/437 A61K31/5377 A61K31/538 A61K31/5383 A61P35/00 

Abstract RU 2690663 C2

FIELD: chemistry.

SUBSTANCE: invention relates to organic chemistry and notably to specific imidazo[4,5-c]pyridine derivatives. Invention also relates to a pharmaceutical composition based on a specific imidazo[4,5-c]pyridine derivative useful in treating cancer.

EFFECT: technical result is obtaining novel imidazopyridine derivatives useful as HDM2 protein inhibitors.

17 cl, 1 dwg, 21 tbl, 360 ex

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RU 2 690 663 C2

Authors

Bolisetti Ragkhu

Kammarano Karolin Mishel

Kristofer Mettyu P.

Fradera Linas Fransesk Ksaver

Gkhosh Partkha

Mashasek Mishell

Martines Mishel

Panda Dzhagannatkh

Rojtershan Majkl Khejl

Samala Dzhajya Prakash

Sidzuka Manami

Sun Binyuan

Tompson Kristofer Frensis

Toni Kurisseri Antkhappan

Trotter B. Uesli

Voss Mettyu E.

Yan Lipin

Altman Majkl D.

Bodzhen Stefan L.

Doll Ronald Dzh.

Dates

2019-06-05Published

2013-12-18Filed