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2 693 404

(13)

(51)

IPC

C07D401/14(2006-01-01)

C07D401/10(2006-01-01)

C07D405/14(2006-01-01)

A61K31/4709(2006-01-01)

A61P35/00(2006-01-01)

A61P37/00(2006-01-01)

(21) (22)

Application

2016106002, 2014-07-22

(24)

Start date

2014-07-22

(22)

Actual filing date

2014-07-22

(45)

Published

2019-07-02

(72)

Inventor

Kasara PatrikLe-Digore TerriAnlen Zhan-MishelStark Zherom-BenuaLe-Tiran ArnoDe-Nantej GijomZhanest OliveDejvidson Dzhejms Eduard PolMarri Dzhejms BrukChen ItszenUolmsli KlerGrem Kristofer DzhonRej StyuartMaddoks DanielBedford Sajmon

(73)

Holder

Le Laboratuar ServeVernalis Limited

NOVEL INDOLE AND PYRROLE COMPOUNDS, A METHOD FOR PRODUCTION THEREOF AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Russian patent published in 2019 - IPC C07D401/14 C07D401/10 C07D405/14 A61K31/4709 A61P35/00 A61P37/00

Abstract RU 2693404 C2

FIELD: pharmaceuticals.

SUBSTANCE: invention relates to novel compounds of formula (I), as well as to pharmaceutical compositions based thereon and use.

EFFECT: obtaining novel compounds, as well as pharmaceutical compositions having Bcl-2 inhibitory activity, suitable for treating mediated diseases, such as cancer, autoimmune diseases.

19 cl, 211 ex, 2 tbl

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RU 2 693 404 C2

Authors

Kasara Patrik

Le-Digore Terri

Anlen Zhan-Mishel

Stark Zherom-Benua

Le-Tiran Arno

De-Nantej Gijom

Zhanest Olive

Dejvidson Dzhejms Eduard Pol

Marri Dzhejms Bruk

Chen Itszen

Uolmsli Kler

Grem Kristofer Dzhon

Rej Styuart

Maddoks Daniel

Bedford Sajmon

Dates

2019-07-02—Published

2014-07-22—Filed