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(19)

RU

(11)

2 760 554

(13)

C1

(51)

IPC

C07D209/12(2006-01-01)

C07D307/80(2006-01-01)

C07D307/81(2006-01-01)

C07D333/56(2006-01-01)

C07D403/12(2006-01-01)

C07D405/04(2006-01-01)

C07D405/12(2006-01-01)

C07D409/12(2006-01-01)

C07D471/04(2006-01-01)

C07D487/04(2006-01-01)

C07D491/04(2006-01-01)

C07D495/04(2006-01-01)

A61K31/381(2006-01-01)

A61K31/4355(2006-01-01)

A61K31/437(2006-01-01)

A61P35/00(2006-01-01)

(21) (22)

Application

2018102368, 2016-06-22

(24)

Start date

2016-06-22

(22)

Actual filing date

2016-06-22

(45)

Published

2021-11-29

(72)

Inventor

Balint BalazhChekej MartonSabo ZoltanSlavik ZoltanKochi AndrashShanrion MajyaZhenest OliveChen ItszenDejvidson Dzhejms Eduard PolMyurrej Dzhejms BrukShiposh SabolchOndi LeventeProsenyak Agnesh

(73)

Holder

Le Laboratuar ServeVernalis Limited

NEW BICYCLIC DERIVATIVES, METHOD FOR THEIR PRODUCTION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM Russian patent published in 2021 - IPC C07D209/12 C07D307/80 C07D307/81 C07D333/56 C07D403/12 C07D405/04 C07D405/12 C07D409/12 C07D471/04 C07D487/04 C07D491/04 C07D495/04 A61K31/381 A61K31/4355 A61K31/437 A61P35/00 

Abstract RU 2760554 C1

FIELD: pharmaceutics.

SUBSTANCE: invention relates to bicyclic derivatives of the formula (I), where R1, R2, R3, R4, R5, R6, R7, R8, R14, W, А and n are such as defined in the description, to a method for their production and to pharmaceutical composition containing them.

EFFECT: compounds of the present invention are new and have very valuable pharmacological characteristics in the field of apoptosis and oncology.

40 cl, 104 ex, 2 tbl

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RU 2 760 554 C1

Authors

Balint Balazh

Chekej Marton

Sabo Zoltan

Slavik Zoltan

Kochi Andrash

Shanrion Majya

Zhenest Olive

Chen Itszen

Dejvidson Dzhejms Eduard Pol

Myurrej Dzhejms Bruk

Shiposh Sabolch

Ondi Levente

Prosenyak Agnesh

Dates

2021-11-29—Published

2016-06-22—Filed

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