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(19)

RU

(11)

2 703 273

(13)

C2

(51)

IPC

C07D513/04(2006-01-01)

A61K31/519(2006-01-01)

A61P25/00(2006-01-01)

(21) (22)

Application

2016115487, 2014-10-08

(24)

Start date

2014-10-08

(22)

Actual filing date

2014-10-08

(45)

Published

2019-10-16

(72)

Inventor

Yuj TszyanU GoshenYuen Po-VajVillemur EliziyaShvarts YakobLi KuonSellers BendzhaminVolgraf Metyu

(73)

Holder

F. Hoffmann-La Roche Ag

THIAZOLOPYRIMIDINONES AS MODULATORS OF NMDA RECEPTOR ACTIVITY Russian patent published in 2019 - IPC C07D513/04 A61K31/519 A61P25/00 

Abstract RU 2703273 C2

FIELD: chemistry.

SUBSTANCE: invention relates to thiazolopyrimidinone compounds of formula (II) and pharmaceutical compositions based thereon.

EFFECT: technical result is obtaining novel compounds which can be used as a drug exhibiting activity of NR2A-selective modulation of NMDA receptor.

67 cl, 3 tbl, 267 ex

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RU 2 703 273 C2

Authors

Yuj Tszyan

U Goshen

Yuen Po-Vaj

Villemur Eliziya

Shvarts Yakob

Li Kuon

Sellers Bendzhamin

Volgraf Metyu

Dates

2019-10-16—Published

2014-10-08—Filed

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