IMIDAZOPYRROLOPYRINE DERIVATIVES USEFUL FOR TREATING DISEASES CAUSED BY ABNORMAL ACTIVITY OF PROTEIN KINASES JAK1, JAK3 OR SYK Russian patent published in 2020 - IPC C07D471/14 C07D487/14 A61K31/437 A61K31/4985 A61P37/06 A61P11/06 A61P25/28 

Abstract RU 2711869 C2

FIELD: chemistry.

SUBSTANCE: invention relates to organic chemistry and specifically to a compound of the structure given below and a pharmaceutically acceptable salt thereof.

EFFECT: technical result is obtaining a novel heterocyclic compound useful for treating various pathological conditions mediated by abnormal activity of kinases of JAK family, and in particular for treating rheumatoid arthritis.

1 cl, 54 tbl, 690 ex

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RU 2 711 869 C2

Authors

Vishart Nil

Ardzhiriadi Mariya A.

Koldervud Devid Dzh.

Eriksson Anna M.

Fyamengo Brajan A.

Frenk Kristin E.

Fridman Majkl

Dzhorzh Don M.

Godken Erik R.

Dzhozefson Natan S.

Li Bitsin S.

Morytko Majkl Dzh.

Styuart Kent D.

Voss Dzheffri V.

Uollejs Grir A.

Van Lu

Voller Kevin R.

Dates

2020-01-22Published

2010-12-01Filed